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Tazemetostat hydrobromide

Glpbio
Catalog No:GC38163-10mM (in 1mL DMSO) CAS No.:1467052-75-0 MDLNo: Brand:Glpbio purity: 特性: Purpose:Tazemetostat hydrobromide (EPZ-6438 hydrobromide) 是一种有效,选择性,口服的 EZH2 抑制剂。Tazemetostat hydrobromide 抑制含有 PRC2 复合体的野生型 EZH2 的活性, Ki 值为 2.5±0.5 nM。Tazemetostat hydrobromide 抑制 EZH2,在肽测定和核小体测定中 IC50 分别为 11 和 16 nM。Tazemetostat hydrobromide 抑制大鼠 EZH2,IC50 为 4 nM。Tazemetostat hydrobromide 还抑制 EZH1,IC50 为 392 nM。DMSO: 100 mg/mL (152.99 mM)
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